Compile Data Set for Download or QSAR
maximum 50k data
Found 49 of ic50 data for polymerid = 9920,49000281,50002318,50003238
TargetSodium/potassium-transporting ATPase subunit alpha-1(Canis familiaris)
University Of Manitoba

Curated by ChEMBL
LigandPNGBDBM46356(DIGITOXIN | MLS000069787 | SMR000058529 | US106680...)
Affinity DataIC50:  8nMAssay Description:Inhibition of [3H]ouabain binding to Digitalis receptor in dog heart microsomesMore data for this Ligand-Target Pair
TargetSodium/potassium-transporting ATPase subunit alpha-1(Canis familiaris)
University Of Manitoba

Curated by ChEMBL
LigandPNGBDBM50408112(CHEMBL2069115)
Affinity DataIC50:  8.30nMAssay Description:Inhibition of [3H]ouabain binding to Digitalis receptor in dog heart microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/potassium-transporting ATPase subunit alpha-1(Canis familiaris)
University Of Manitoba

Curated by ChEMBL
LigandPNGBDBM50408116(CHEMBL2069118)
Affinity DataIC50:  13nMAssay Description:Inhibition of [3H]ouabain binding to Digitalis receptor in dog heart microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/potassium-transporting ATPase subunit alpha-1(Canis familiaris)
University Of Manitoba

Curated by ChEMBL
LigandPNGBDBM50408117(CHEMBL2069066)
Affinity DataIC50:  30nMAssay Description:Inhibition of [3H]ouabain binding to Digitalis receptor in dog heart microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/potassium-transporting ATPase subunit alpha-1(Canis familiaris)
University Of Manitoba

Curated by ChEMBL
LigandPNGBDBM50408111(CHEMBL2069075)
Affinity DataIC50:  45.5nMAssay Description:Inhibition of [3H]ouabain binding to Digitalis receptor in dog heart microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/potassium-transporting ATPase subunit alpha-1(Sus scrofa)
Unibioscreen

Curated by ChEMBL
LigandPNGBDBM50161249(3a,11a-dihydroxy-4''-imino-9,15a-dimethyl-1-(5-oxo...)
Affinity DataIC50:  68nMAssay Description:In vitro inhibitory activity against porcine Na+/K+-ATPaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/potassium-transporting ATPase subunit alpha-1(Sus scrofa)
Unibioscreen

Curated by ChEMBL
LigandPNGBDBM50161262(11a-hydroxy-3a,13a-di(hydroxymethyl)-9,15a-dimethy...)
Affinity DataIC50:  75nMAssay Description:In vitro inhibitory activity against porcine Na+/K+-ATPaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/potassium-transporting ATPase subunit alpha-1(Canis familiaris)
University Of Manitoba

Curated by ChEMBL
LigandPNGBDBM50605867(CHEMBL469045)
Affinity DataIC50:  140nMAssay Description:Inhibition of Beagle dog kidney NA+/K+ ATPase alpha 1 by measuring 32P-ATP hydrolysis preincubated for 10 mins followed by addition of 32P-ATP measur...More data for this Ligand-Target Pair
TargetSodium/potassium-transporting ATPase subunit alpha-1(Canis familiaris)
University Of Manitoba

Curated by ChEMBL
LigandPNGBDBM50408276(CHEMBL2068996)
Affinity DataIC50:  160nMAssay Description:Inhibition of Na+/K+ ATPase from dog kidneyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/potassium-transporting ATPase subunit alpha-1(Canis familiaris)
University Of Manitoba

Curated by ChEMBL
LigandPNGBDBM50408114(CHEMBL2069070)
Affinity DataIC50:  230nMAssay Description:Inhibition of [3H]ouabain binding to Digitalis receptor in dog heart microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/potassium-transporting ATPase subunit alpha-1(Canis familiaris)
University Of Manitoba

Curated by ChEMBL
LigandPNGBDBM50408439(CHEMBL2068890)
Affinity DataIC50:  250nMAssay Description:In vitro inhibitory concentration against dog kidney Na+,K+-ATPaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/potassium-transporting ATPase subunit alpha-1(Homo sapiens (Human))
Universidade Federal De S£O Jo£O Del Rei

Curated by ChEMBL
LigandPNGBDBM46355(DIGOXIN | MLS000069819 | SMR000059217 | US10668094...)
Affinity DataIC50:  290nMAssay Description:Inhibition of human kidney Na(+)/K(+) ATPase alpha-1 assessed as amount of Pi release after 1 hr by colorimetric methodMore data for this Ligand-Target Pair
TargetSodium/potassium-transporting ATPase subunit alpha-1(Canis familiaris)
University Of Manitoba

Curated by ChEMBL
LigandPNGBDBM50408921(CHEMBL2068972)
Affinity DataIC50:  320nMAssay Description:In vitro inhibitory concentration against dog kidney Na+,K+-ATPaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/potassium-transporting ATPase subunit alpha-1(Homo sapiens (Human))
Universidade Federal De S£O Jo£O Del Rei

Curated by ChEMBL
LigandPNGBDBM50096255(CHEMBL3594278)
Affinity DataIC50:  340nMAssay Description:Inhibition of human kidney Na(+)/K(+) ATPase alpha-1 assessed as amount of Pi release after 1 hr by colorimetric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/potassium-transporting ATPase subunit alpha-1(Canis familiaris)
University Of Manitoba

Curated by ChEMBL
LigandPNGBDBM46355(DIGOXIN | MLS000069819 | SMR000059217 | US10668094...)
Affinity DataIC50:  500nMAssay Description:In vitro inhibitory concentration against dog kidney Na+,K+-ATPaseMore data for this Ligand-Target Pair
TargetSodium/potassium-transporting ATPase subunit alpha-1(Canis familiaris)
University Of Manitoba

Curated by ChEMBL
LigandPNGBDBM66977(3-[(3S,5R,8R,9S,10S,13R,14S,17R)-10,13-dimethyl-3,...)
Affinity DataIC50:  500nMAssay Description:In vitro inhibitory concentration against dog kidney Na+,K+-ATPaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/potassium-transporting ATPase subunit alpha-1(Canis familiaris)
University Of Manitoba

Curated by ChEMBL
LigandPNGBDBM46355(DIGOXIN | MLS000069819 | SMR000059217 | US10668094...)
Affinity DataIC50:  500nMAssay Description:Inhibition of Na+/K+ ATPase from dog kidneyMore data for this Ligand-Target Pair
TargetSodium/potassium-transporting ATPase subunit alpha-1(Canis familiaris)
University Of Manitoba

Curated by ChEMBL
LigandPNGBDBM66977(3-[(3S,5R,8R,9S,10S,13R,14S,17R)-10,13-dimethyl-3,...)
Affinity DataIC50:  500nMAssay Description:Inhibition of Na+/K+ ATPase from dog kidneyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/potassium-transporting ATPase subunit alpha-1(Homo sapiens (Human))
Universidade Federal De S£O Jo£O Del Rei

Curated by ChEMBL
LigandPNGBDBM50096254(CHEMBL3594276)
Affinity DataIC50:  570nMAssay Description:Inhibition of human kidney Na(+)/K(+) ATPase alpha-1 assessed as amount of Pi release after 1 hr by colorimetric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/potassium-transporting ATPase subunit alpha-1(Canis familiaris)
University Of Manitoba

Curated by ChEMBL
LigandPNGBDBM50408115(CHEMBL2069067)
Affinity DataIC50:  660nMAssay Description:Inhibition of [3H]ouabain binding to Digitalis receptor in dog heart microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/potassium-transporting ATPase subunit alpha-1(Canis familiaris)
University Of Manitoba

Curated by ChEMBL
LigandPNGBDBM50408917(CHEMBL2068902)
Affinity DataIC50:  1.25E+3nMAssay Description:In vitro inhibitory concentration against dog kidney Na+,K+-ATPaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/potassium-transporting ATPase subunit alpha-1(Canis familiaris)
University Of Manitoba

Curated by ChEMBL
LigandPNGBDBM50408275(CHEMBL2068885)
Affinity DataIC50:  1.58E+3nMAssay Description:Inhibition of Na+/K+ ATPase from dog kidneyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/potassium-transporting ATPase subunit alpha-1(Canis familiaris)
University Of Manitoba

Curated by ChEMBL
LigandPNGBDBM50408916(CHEMBL2068975)
Affinity DataIC50:  1.58E+3nMAssay Description:In vitro inhibitory concentration against dog kidney Na+,K+-ATPaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/potassium-transporting ATPase subunit alpha-1(Sus scrofa)
Unibioscreen

Curated by ChEMBL
LigandPNGBDBM50161244(CHEMBL369515 | Uscharin derivative)
Affinity DataIC50:  1.89E+3nMAssay Description:In vitro inhibitory activity against porcine Na+/K+-ATPaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/potassium-transporting ATPase subunit alpha-1(Canis familiaris)
University Of Manitoba

Curated by ChEMBL
LigandPNGBDBM50408119(CHEMBL2069069)
Affinity DataIC50:  1.89E+3nMAssay Description:Inhibition of [3H]ouabain binding to Digitalis receptor in dog heart microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/potassium-transporting ATPase subunit alpha-1(Canis familiaris)
University Of Manitoba

Curated by ChEMBL
LigandPNGBDBM50408282(CHEMBL2069057)
Affinity DataIC50:  2.00E+3nMAssay Description:Inhibition of Na+/K+ ATPase from dog kidneyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/potassium-transporting ATPase subunit alpha-1(Canis familiaris)
University Of Manitoba

Curated by ChEMBL
LigandPNGBDBM50408113(CHEMBL2069072)
Affinity DataIC50:  2.20E+3nMAssay Description:Inhibition of [3H]ouabain binding to Digitalis receptor in dog heart microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/potassium-transporting ATPase subunit alpha-1(Canis familiaris)
University Of Manitoba

Curated by ChEMBL
LigandPNGBDBM50408281(CHEMBL2068935 | CHEMBL2068940)
Affinity DataIC50:  2.50E+3nMAssay Description:Inhibition of Na+/K+ ATPase from dog kidneyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/potassium-transporting ATPase subunit alpha-1(Canis familiaris)
University Of Manitoba

Curated by ChEMBL
LigandPNGBDBM50408118(CHEMBL2069074)
Affinity DataIC50:  3.22E+3nMAssay Description:Inhibition of [3H]ouabain binding to Digitalis receptor in dog heart microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/potassium-transporting ATPase subunit alpha-1(Canis familiaris)
University Of Manitoba

Curated by ChEMBL
LigandPNGBDBM50408279(CHEMBL2069128)
Affinity DataIC50:  3.98E+3nMAssay Description:Inhibition of Na+/K+ ATPase from dog kidneyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/potassium-transporting ATPase subunit alpha-1(Sus scrofa)
Unibioscreen

Curated by ChEMBL
LigandPNGBDBM50161268(CHEMBL366906 | Uscharin derivative)
Affinity DataIC50:  4.08E+3nMAssay Description:In vitro inhibitory activity against porcine Na+/K+-ATPaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/potassium-transporting ATPase subunit alpha-1(Canis familiaris)
University Of Manitoba

Curated by ChEMBL
LigandPNGBDBM50408120(CHEMBL2069071)
Affinity DataIC50:  4.73E+3nMAssay Description:Inhibition of [3H]ouabain binding to Digitalis receptor in dog heart microsomesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/potassium-transporting ATPase subunit alpha-1(Canis familiaris)
University Of Manitoba

Curated by ChEMBL
LigandPNGBDBM50408280(CHEMBL2068992)
Affinity DataIC50:  5.00E+3nMAssay Description:Inhibition of Na+/K+ ATPase from dog kidneyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/potassium-transporting ATPase subunit alpha-1(Canis familiaris)
University Of Manitoba

Curated by ChEMBL
LigandPNGBDBM50408920(CHEMBL2069058)
Affinity DataIC50:  6.30E+3nMAssay Description:In vitro inhibitory concentration against dog kidney Na+,K+-ATPaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/potassium-transporting ATPase subunit alpha-1(Canis familiaris)
University Of Manitoba

Curated by ChEMBL
LigandPNGBDBM50408278(CHEMBL2068942)
Affinity DataIC50:  6.31E+3nMAssay Description:Inhibition of Na+/K+ ATPase from dog kidneyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/potassium-transporting ATPase subunit alpha-1(Canis familiaris)
University Of Manitoba

Curated by ChEMBL
LigandPNGBDBM50408281(CHEMBL2068935 | CHEMBL2068940)
Affinity DataIC50:  6.31E+3nMAssay Description:Inhibition of Na+/K+ ATPase from dog kidneyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/potassium-transporting ATPase subunit alpha-1(Canis familiaris)
University Of Manitoba

Curated by ChEMBL
LigandPNGBDBM50408277(CHEMBL2068936)
Affinity DataIC50:  7.94E+3nMAssay Description:Inhibition of Na+/K+ ATPase from dog kidneyMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/potassium-transporting ATPase subunit alpha-1(RAT)
Albert-Ludwigs-University Of Freiburg

Curated by ChEMBL
LigandPNGBDBM50409816(ABAMECTIN)
Affinity DataIC50:  8.23E+3nMAssay Description:Inhibition of Wistar rat kidney Na+,K+-ATPase alpha1 after 2 hrsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/potassium-transporting ATPase subunit alpha-1(Homo sapiens (Human))
Universidade Federal De S£O Jo£O Del Rei

Curated by ChEMBL
LigandPNGBDBM50096256(CHEMBL3594279)
Affinity DataIC50:  9.80E+3nMAssay Description:Inhibition of human kidney Na(+)/K(+) ATPase alpha-1 assessed as amount of Pi release after 1 hr by colorimetric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/potassium-transporting ATPase subunit alpha-1(Homo sapiens (Human))
Universidade Federal De S£O Jo£O Del Rei

Curated by ChEMBL
LigandPNGBDBM50096257(CHEMBL3594280)
Affinity DataIC50:  1.10E+4nMAssay Description:Inhibition of human kidney Na(+)/K(+) ATPase alpha-1 assessed as amount of Pi release after 1 hr by colorimetric methodMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/potassium-transporting ATPase subunit alpha-1(Sus scrofa)
Unibioscreen

Curated by ChEMBL
LigandPNGBDBM50161245(11a-hydroxy-3a-hydroxymethyl-4''-imino-9,15a-dimet...)
Affinity DataIC50:  1.21E+4nMAssay Description:In vitro inhibitory activity against porcine Na+/K+-ATPaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/potassium-transporting ATPase subunit alpha-1(Canis familiaris)
University Of Manitoba

Curated by ChEMBL
LigandPNGBDBM50408915(CHEMBL2068981)
Affinity DataIC50:  2.50E+4nMAssay Description:In vitro inhibitory concentration against dog kidney Na+,K+-ATPaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/potassium-transporting ATPase subunit alpha-1(Canis familiaris)
University Of Manitoba

Curated by ChEMBL
LigandPNGBDBM50408914(CHEMBL2068977)
Affinity DataIC50:  4.00E+4nMAssay Description:In vitro inhibitory concentration against dog kidney Na+,K+-ATPaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/potassium-transporting ATPase subunit alpha-1(Sus scrofa)
Unibioscreen

Curated by ChEMBL
LigandPNGBDBM50161253(CHEMBL426228 | Uscharin derivative)
Affinity DataIC50: >5.00E+4nMAssay Description:In vitro inhibitory activity against porcine Na+/K+-ATPaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/potassium-transporting ATPase subunit alpha-1(Sus scrofa)
Unibioscreen

Curated by ChEMBL
LigandPNGBDBM50161252(CHEMBL427124 | Uscharin derivative)
Affinity DataIC50:  5.00E+4nMAssay Description:In vitro inhibitory activity against porcine Na+/K+-ATPaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/potassium-transporting ATPase subunit alpha-1(Sus scrofa)
Unibioscreen

Curated by ChEMBL
LigandPNGBDBM50161272(CHEMBL262795 | Uscharin derivative)
Affinity DataIC50: >5.00E+4nMAssay Description:In vitro inhibitory activity against porcine Na+/K+-ATPaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/potassium-transporting ATPase subunit alpha-1(Sus scrofa)
Unibioscreen

Curated by ChEMBL
LigandPNGBDBM50161246(11a-hydroxy-3a-hydroxymethyl-4''-imino-9,15a-dimet...)
Affinity DataIC50: >5.00E+4nMAssay Description:In vitro inhibitory activity against porcine Na+/K+-ATPaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/potassium-transporting ATPase subunit alpha-1(Canis familiaris)
University Of Manitoba

Curated by ChEMBL
LigandPNGBDBM50408918(CHEMBL2068898 | CHEMBL2068976)
Affinity DataIC50:  1.00E+5nMAssay Description:In vitro inhibitory concentration against dog kidney Na+,K+-ATPaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetSodium/potassium-transporting ATPase subunit alpha-1(Canis familiaris)
University Of Manitoba

Curated by ChEMBL
LigandPNGBDBM50408918(CHEMBL2068898 | CHEMBL2068976)
Affinity DataIC50: >1.00E+5nMAssay Description:In vitro inhibitory concentration against dog kidney Na+,K+-ATPaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed